SCHEMBL6962052

SCHEMBL6962052

COc1ccc2cc(/C(C)=C\C(=O)O)ccc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.65
CYP1A2 P05177 3/20 0.55
ALDH1A1 P00352 2/20 0.55
HPGD P15428 1/20 0.55
CYP2C19 P33261 1/20 0.55
HSD17B10 Q99714 1/20 0.55
NPC1 O15118 3/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
PLAU P00749 1/20 0.48
AKR1C3 P42330 4/20 0.47
AKR1C2 P52895 4/20 0.47
PTGS1 P23219 3/20 0.47
PTGS2 P35354 3/20 0.46
CDC42 P60953 1/20 0.46
RAC1 P63000 1/20 0.46
TSHR P16473 1/20 0.46
SLC22A6 Q4U2R8 1/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962058 1.00 KDM4E (0.65) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL6962047 1.00 KDM4E (0.65) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
Hydrochloric Acid SCHEMBL6785127 0.98 KDM4E (0.63) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL11739013 0.89 KDM4E (0.62) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL11157055 0.89 KDM4E (0.62) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL12900045 0.86 KDM4E (0.58) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL28613089 0.86 KDM4E (0.58) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL986740 0.86 KDM4E (0.58) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL6785122 0.86 KDM4E (0.58) KDM4ECYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL986741 0.86 KDM4E (0.58) KDM4ECYP1A2ALDH1A1HPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed
US-4420639-A Aromatic compounds BEECHAM GROUP LIMITED (GB) 1983-12-13 US disclosed