SCHEMBL696244

SCHEMBL696244

O=C(Nc1ccn(Cc2c(F)cccc2C(F)(F)F)n1)c1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STIM1 Q13586 2/20 0.80
ORAI1 Q96D31 2/20 0.80
NPC1 O15118 5/20 0.57
RAB9A P51151 5/20 0.57
ALDH1A1 P00352 4/20 0.57
SMN1; SMN2 Q16637 10/20 0.57
NFKB1 P19838 1/20 0.57
NFKB2 Q00653 1/20 0.57
RELA Q04206 1/20 0.57
LMNA P02545 7/20 0.57
ORAI3 Q9BRQ5 1/20 0.56
EGFR P00533 1/20 0.50
NPSR1 Q6W5P4 3/20 0.48
HTT P42858 2/20 0.48
TSHR P16473 1/20 0.48
MAPT P10636 3/20 0.48
STAT3 P40763 2/20 0.47
HPGD P15428 1/20 0.47
PKM P14618 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL759169 0.89 STIM1 (0.80) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL715052 0.89 STIM1 (1.00) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL30096538 0.89 STIM1 (1.00) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL756322 0.86 STIM1 (0.86) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL755899 0.85 STIM1 (0.74) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL757813 0.85 STIM1 (0.74) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL758373 0.81 STIM1 (0.68) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL758374 0.81 STIM1 (0.84) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL760683 0.79 STIM1 (0.78) STIM1ORAI1NPC1RAB9AALDH1A1
SCHEMBL759947 0.79 STIM1 (0.79) STIM1ORAI1NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421835-A1 N-PYRAZOLYL CARBOXAMIDES AS CRAC CHANNEL INHIBITORS Glaxo Group Limited (GB) 2012-02-29 EP disclosed