SCHEMBL6964780

SCHEMBL6964780

CCN1c2ncc(C#Cc3ccccn3)cc2C(=O)N(C)c2cccnc21

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPC1 O15118 1/20 0.39
HCRTR1 O43613 1/20 0.39
RAB9A P51151 1/20 0.39
POLB P06746 1/20 0.39
PTPN7 P35236 1/20 0.39
DUSP3 P51452 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
GRM5 P41594 5/20 0.39
BRD4 O60885 6/20 0.37
RIPK1 Q13546 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955026 0.91 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19GRM5BRD4
SCHEMBL6954952 0.87 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19GRM5BRD4
SCHEMBL6965781 0.84 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19GRM5BRD4
SCHEMBL6952762 0.84 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19BRD4
SCHEMBL8299587 0.78 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19BRD4
SCHEMBL6959985 0.78 CYP3A4 (0.53) CYP3A4CYP2C9CYP2C19BRD4
SCHEMBL6956040 0.78 CYP3A4 (0.53) CYP3A4CYP2C9CYP2C19BRD4
SCHEMBL5745003 0.78 CYP3A4 (0.53) CYP3A4CYP2C9CYP2C19BRD4
SCHEMBL6961652 0.78 CYP2C9 (0.53) CYP3A4CYP2C9CYP2C19POLBGRM5
SCHEMBL6961657 0.78 CYP2C9 (0.53) CYP3A4CYP2C9CYP2C19POLBGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767172-B1 8-Arylalkyl- and 8-arylheteroalkyl-5, 11-dihydro-6H-dipyrido-[3,2-b:2', 3'-e][1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMA (US) 2003-03-26 EP disclosed
US-5705499-A VIRICIDES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1998-01-06 US disclosed
EP-0767172-A1 8-Arylalkyl- and 8-arylheteroalkyl-5, 11-dihydro-6H-dipyrido-[3,2-b:2', 3'-e][1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1997-04-09 EP disclosed