SCHEMBL6965003

SCHEMBL6965003

CCCc1nc(OC)c(NC(=S)N2CCN(c3cc(C)cc(C)c3)CC2)cc1C

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 7/20 0.51
CYP3A4 P08684 3/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
PKM P14618 1/20 0.45
NPC1 O15118 2/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958260 0.91 PHGDH (0.55) PHGDHCYP3A4CYP2C19MEN1KMT2A
SCHEMBL6956612 0.89 PHGDH (0.40) PHGDHCYP3A4MEN1KMT2APOLB
SCHEMBL6657881 0.86 PHGDH (0.56) PHGDHCYP3A4CYP2C19MEN1KMT2A
SCHEMBL6953108 0.85 GAA (0.51) PHGDHCYP3A4CYP2C19MEN1KMT2A
SCHEMBL6653887 0.82 PHGDH (0.52) PHGDHCYP3A4CYP2C19MEN1KMT2A
SCHEMBL6651807 0.82 MAPT (0.48) PHGDHCYP3A4CYP2C19MEN1KMT2A
SCHEMBL6959667 0.80 PHGDH (0.42) PHGDHCYP3A4MEN1KMT2APOLB
SCHEMBL6956121 0.80 KMT2A (0.45) PHGDHCYP3A4CYP2C19MEN1KMT2A
SCHEMBL5395201 0.79 HCAR2 (0.40) PHGDHMEN1KMT2ALMNAALDH1A1
SCHEMBL6651512 0.78 PHGDH (0.52) PHGDHCYP3A4CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850222-B1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARM CO LTD (KR) 2003-05-28 EP disclosed
US-6028195-A AN ANTITUMOR AGENT WITH VERY LOW TOXICITIES SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-02-22 US disclosed