SCHEMBL6970657

SCHEMBL6970657

Cc1ccc2c(c1)NC(=O)CCN2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.49
MMP12 P39900 1/20 0.47
PARP10 Q53GL7 2/20 0.45
PARP11 Q9NR21 1/20 0.45
PARP1 P09874 1/20 0.45
BRD4 O60885 1/20 0.43
CREBBP Q92793 1/20 0.43
CSNK1G1 Q9HCP0 1/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 3/20 0.42
GAA P10253 2/20 0.42
HSD17B10 Q99714 1/20 0.42
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
NPC1 O15118 1/20 0.41
CYP2C9 P11712 1/20 0.41
MCL1 Q07820 1/20 0.41
CRBN Q96SW2 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960230 0.93 EPHX2 (0.49) EPHX2MMP12PARP10PARP11PARP1
SCHEMBL30509208 0.81 EPHX2 (0.51) EPHX2MMP12BRD4CREBBPCSNK1G1
SCHEMBL11455059 0.81 EPHX2 (0.51) EPHX2MMP12BRD4CREBBPCSNK1G1
SCHEMBL19203466 0.79 CA9 (0.59) ALDH1A1MAPTGAASMN1; SMN2NPC1
SCHEMBL29126120 0.79 PARP1 (0.45) PARP10PARP1MAPTSMN1; SMN2CYP1A2
SCHEMBL30697324 0.79 PARP1 (0.45) PARP10PARP1MAPTSMN1; SMN2CYP1A2
SCHEMBL6959254 0.79 AHR (0.51) PARP10PARP1MAPTCYP1A2CYP2C19
SCHEMBL30832124 0.79 CMA1 (0.51) PARP10PARP11PARP1BRD4CRBN
SCHEMBL6968312 0.78 PDE3B (0.53) ALDH1A1MAPTCYP1A2CYP2C19NPC1
SCHEMBL10274620 0.77 EPHX2 (0.55) EPHX2MMP12BRD4CREBBPCSNK1G1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed