SCHEMBL6971666

SCHEMBL6971666

CC(=O)OCCN1[CH]CNCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
SLC18A3 Q16572 1/20 0.38
CHRM5 P08912 2/20 0.32
CHRM1 P11229 2/20 0.32
CHRM3 P20309 2/20 0.32
PGR P06401 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
HTR1A P08908 1/20 0.32
CHRNB2 P17787 1/20 0.32
TBXA2R P21731 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA7 P36544 1/20 0.32
CHRNA4 P43681 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CHRNA10 Q9GZZ6 1/20 0.32
CHRNA9 Q9UGM1 1/20 0.32
TSHR P16473 1/20 0.32
ADORA2B P29275 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1476931 0.78 MEN1 (0.34) ALDH1A1MEN1KMT2A
SCHEMBL5953471 0.74 SLC18A3 (0.49) ALDH1A1SLC18A3CHRM5CHRM3SMN1; SMN2
SCHEMBL6971664 0.74 SLC18A3 (0.49) ALDH1A1SLC18A3CHRM5CHRM3SMN1; SMN2
SCHEMBL7344795 0.73 GLA (0.35) SMN1; SMN2MEN1KMT2A
Hydrochloric Acid SCHEMBL7421281 0.73 SLC18A3 (0.48) ALDH1A1SLC18A3CHRM5CHRM3GAA
Hydrochloric Acid SCHEMBL6498838 0.73 SLC18A3 (0.48) ALDH1A1SLC18A3CHRM5CHRM3GAA
SCHEMBL9061088 0.71 SLC18A3 (0.43) ALDH1A1SLC18A3CHRM5CHRM1CHRM3
SCHEMBL3044885 0.71
SCHEMBL28024374 0.69 CXCR4 (0.49) ALDH1A1SLC18A3CHRM5CHRM3MEN1
SCHEMBL3533333 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed