SCHEMBL697178

SCHEMBL697178

CC(=O)c1cccc(Oc2ccc(C(=O)COC(=O)[C@@H]3CCCN3C(=O)OC(C)(C)C)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.50
HRH2 P25021 1/20 0.44
HRH1 P35367 1/20 0.44
UCHL1 P09936 3/20 0.43
FKBP1A P62942 2/20 0.43
EPHX2 P34913 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
KLK7 P49862 1/20 0.41
LMNA P02545 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
USP30 Q70CQ3 2/20 0.40
PARP10 Q53GL7 2/20 0.40
ALDH1A1 P00352 1/20 0.40
GFER P55789 1/20 0.40
PARP14 Q460N5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204107 0.95 NPC1 (0.46) NPC1HRH2HRH1UCHL1FKBP1A
SCHEMBL564404 0.95 NPC1 (0.46) NPC1HRH2HRH1UCHL1FKBP1A
SCHEMBL2706083 0.90 NPC1 (0.52) NPC1HRH2HRH1UCHL1EPHX2
SCHEMBL203942 0.90 NPC1 (0.52) NPC1HRH2HRH1UCHL1EPHX2
SCHEMBL15481363 0.87 NPC1 (0.41) NPC1HRH2HRH1UCHL1FKBP1A
SCHEMBL18213987 0.85 NPC1 (0.60) NPC1HRH2HRH1UCHL1EPHX2
SCHEMBL18209654 0.85 NPC1 (0.60) NPC1HRH2HRH1UCHL1EPHX2
SCHEMBL4955279 0.85 KLK7 (0.53) NPC1UCHL1FKBP1AEPHX2MEN1
SCHEMBL15848456 0.85 KLK7 (0.53) NPC1UCHL1FKBP1AEPHX2MEN1
SCHEMBL15848455 0.85 KLK7 (0.53) NPC1UCHL1FKBP1AEPHX2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421855-A1 DIARYL ETHERS Tibotec Pharmaceuticals (IE) 2012-02-29 EP disclosed
WO-2010122162-A1 DIARYL ETHERS TIBOTEC PHARMACEUTICALS (IE) 2010-10-28 WO disclosed