SCHEMBL6972472

SCHEMBL6972472

COC(=O)CCNC1CCC1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.57
TSHR P16473 3/20 0.46
CA12 O43570 3/20 0.44
CA14 Q9ULX7 3/20 0.44
NPSR1 Q6W5P4 2/20 0.39
VCP P55072 1/20 0.39
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL619500 0.96 EPHX2 (0.62) EPHX2TSHRCA12CA14NPSR1
SCHEMBL1202915 0.94 EPHX2 (0.65) EPHX2TSHRCA12CA14NPSR1
SCHEMBL12931771 0.94 EPHX2 (0.65) EPHX2TSHRCA12CA14NPSR1
SCHEMBL16473262 0.94 EPHX2 (0.65) EPHX2TSHRCA12CA14NPSR1
SCHEMBL9805865 0.92 EPHX2 (0.51) EPHX2TSHRCA12CA14VCP
Hydrochloric Acid SCHEMBL7295649 0.90 EPHX2 (0.50) EPHX2TSHRCA12CA14VCP
SCHEMBL3649522 0.85 EPHX2 (0.64) EPHX2TSHRKDM4ESMN1; SMN2ALDH1A1
SCHEMBL22927034 0.83 EPHX2 (0.45) EPHX2TSHRCA12CA14VCP
SCHEMBL11288210 0.83 EPHX2 (0.45) EPHX2TSHRCA12CA14VCP
SCHEMBL3667582 0.83 SMYD3 (0.44) EPHX2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110546145-A Azaaryl derivative, preparation method and pharmaceutical application thereof ABBISKO THERAPEUTICS CO LTD 2019-12-06 CN disclosed
EP-1021411-B1 BENZAMIDE DERIVATIVES AS THROMBIN INHIBITORS GLAXO GROUP LTD (GB) 2003-03-05 EP disclosed
US-6326386-B1 ANTICOAGULANT GLAXO GROUP LIMITED (GB) 2001-12-04 US disclosed
EP-1021411-A1 BENZAMIDE DERIVATIVES AS THROMBIN INHIBITORS GLAXO GROUP LIMITED (GB) 2000-07-26 EP disclosed
WO-1997022589-A1 BENZAMIDE DERIVATIVES AS THROMBIN INHIBITORS GLAXO GROUP LIMITED (GB) 1997-06-26 WO disclosed