SCHEMBL6981250

SCHEMBL6981250

Oc1ccc2[nH]cc(-c3ccc(F)cc3)c2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.60
HTR2C P28335 3/20 0.49
CHEK1 O14757 1/20 0.48
WEE1 P30291 1/20 0.48
DYRK1A Q13627 2/20 0.47
TDO2 P48775 6/20 0.46
AR P10275 1/20 0.46
AKR1C3 P42330 1/20 0.46
IDO1 P14902 1/20 0.45
CLK1 P49759 1/20 0.45
CLK2 P49760 1/20 0.45
DYRK2 Q92630 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
HTR1A P08908 2/20 0.44
HTR2A P28223 2/20 0.44
HTR2B P41595 2/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13302269 0.90 DYRK1A (0.55) HTR2CDYRK1ACLK1DYRK2DYRK1B
SCHEMBL9268634 0.86 NR4A2 (0.68) NR4A2TDO2IDO1HTR1AHTR2A
SCHEMBL31140515 0.83 WEE1 (0.49) HTR2CWEE1DYRK1AHTR1AHTR2A
SCHEMBL5435851 0.82 HTR2C (0.56) HTR2CHTR1AHTR2AHTR2BHTR3E
SCHEMBL2361461 0.80 NR4A2 (0.60) NR4A2TDO2HTR1AHTR2AHTR1D
SCHEMBL13302385 0.80 ESR2 (0.49) HTR2CDYRK1ATDO2DYRK2DYRK1B
SCHEMBL9274097 0.80 NR4A2 (0.60) NR4A2DYRK1ATDO2HTR1AHTR2A
SCHEMBL32678326 0.80 NR4A2 (0.60) NR4A2TDO2CLK1HTR1AHTR2A
SCHEMBL32678324 0.80 NR4A2 (0.60) NR4A2TDO2CLK1HTR1AHTR2A
SCHEMBL30954364 0.78 NR4A2 (0.54) NR4A2TDO2IDO1TSHRHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268422-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES Bayer Aktiengesellschaft (DE) 2003-01-02 EP disclosed
WO-2001070687-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES BAYER AKTIENGESELLSCHAFT (DE) 2001-09-27 WO disclosed