SCHEMBL698668

SCHEMBL698668

Cn1c(N2CCC[C@@H]3CCCC[C@@H]32)nc(-c2ccncc2F)cc1=O

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 17/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2D6 P10635 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL697678 1.00 GSK3B (0.54) GSK3BCYP1A2CYP2D6
SCHEMBL698334 1.00 GSK3B (0.54) GSK3BCYP1A2CYP2D6
SCHEMBL697697 1.00 GSK3B (0.54) GSK3BCYP1A2CYP2D6
SCHEMBL696903 0.88 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL697971 0.88 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL697355 0.87 GSK3B (0.61) GSK3BCYP1A2CYP2D6
SCHEMBL697896 0.87 GSK3B (0.61) GSK3BCYP1A2CYP2D6
SCHEMBL8232347 0.87 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL695834 0.87 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL13711312 0.85 GSK3B (0.61) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423207-A2 2-(cyclic amino)-pyrimidone derivatives as TPK1 inhibitors Mitsubishi Tanabe Pharma Corporation (JP) 2012-02-29 EP disclosed