SCHEMBL6989121

SCHEMBL6989121

CC(C)(Nc1cccc(C(=N)N)c1)C(=O)Nc1ccc(-c2ccccc2S(C)(=O)=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
F10 P00742 18/20 0.57
F2 P00734 5/20 0.57
PRSS1 P07477 7/20 0.56
PRSS2 P07478 3/20 0.56
PRSS3 P35030 3/20 0.56
KCNH2 Q12809 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7081758 0.94 PRSS1 (0.59) F10F2PRSS1PRSS2PRSS3
SCHEMBL6995434 0.92 F10 (0.64) F10F2PRSS1PRSS2PRSS3
SCHEMBL6993126 0.89 F10 (0.52) F10F2PRSS1PRSS2PRSS3
Acetic Acid SCHEMBL7080775 0.89 F10 (0.64) F10F2PRSS1PRSS2PRSS3
SCHEMBL6989257 0.89 F10 (0.46) F10F2PRSS1PRSS2PRSS3
Acetic Acid SCHEMBL7080812 0.87 F10 (0.51) F10F2PRSS1PRSS2PRSS3
Trifluoroacetic Acid SCHEMBL7084785 0.84 PRSS1 (0.47) F10F2PRSS1PRSS2PRSS3
SCHEMBL6997959 0.82 F10 (0.52) F10F2PRSS1PRSS2PRSS3
SCHEMBL6224992 0.81 F10 (0.56) F10F2PRSS1PRSS2PRSS3
SCHEMBL7076844 0.81 F10 (0.47) F10F2PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303482-A2 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES MERCK PATENT GmbH (DE) 2003-04-23 EP disclosed
WO-2002008177-A2 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES MERCK PATENT GMBH (DE) 2002-01-31 WO disclosed