SCHEMBL6990890

SCHEMBL6990890

Cc1cc(C)cc(C(=O)Nc2ccc(C(=O)N3CCCCc4sc(Cl)cc43)cc2)c1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 5/20 0.66
AVPR1B P47901 2/20 0.53
NPC1 O15118 1/20 0.51
USP2 O75604 1/20 0.51
ALDH1A1 P00352 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
AVPR2 P30518 1/20 0.51
OXTR P30559 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6991577 0.90 AVPR1A (0.68) AVPR1AAVPR1BRAB9AAVPR2OXTR
SCHEMBL7091449 0.89 AVPR1A (0.65) AVPR1AAVPR1BNPC1ALDH1A1RAB9A
SCHEMBL6994643 0.88 AVPR1A (0.66) AVPR1AAVPR1BRAB9AAVPR2OXTR
SCHEMBL6991357 0.87 AVPR1A (0.68) AVPR1AAVPR1BALDH1A1AVPR2OXTR
SCHEMBL6991936 0.86 AVPR1A (0.67) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL6993363 0.86 AVPR1A (0.67) AVPR1AAVPR1BNPC1RAB9AAVPR2
SCHEMBL6991880 0.86 AVPR1A (0.67) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL6986061 0.85 AVPR1A (0.77) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL6994023 0.85 AVPR1A (0.68) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL6987246 0.84 AVPR1A (0.67) AVPR1AAVPR1BAVPR2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811008-B1 BICYCLIC BENZAZEPINE DERIVATIVES AS VASOPRESSIN ANTAGONISTS WYETH CORP (US) 2003-10-01 EP disclosed