SCHEMBL6993044

SCHEMBL6993044

C[S+]([O-])c1ncc2ncnc(Nc3ccc(-c4ccccc4)cc3)c2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.54
MKNK2 Q9HBH9 2/20 0.50
LMNA P02545 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
RAF1 P04049 2/20 0.40
FLT1 P17948 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPK1 P28482 1/20 0.40
HIF1A Q16665 1/20 0.40
PIK3CA P42336 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6409884 0.93 EGFR (0.62) EGFRMKNK2KDM4EMAPK1
SCHEMBL6996289 0.87 KDR (0.53) EGFRMKNK2LMNANPC1MAPT
SCHEMBL6993198 0.87 EGFR (0.54) EGFRMKNK2
SCHEMBL26696575 0.84 EGFR (0.48) EGFRMKNK2CYP1A2CYP3A4
SCHEMBL6996950 0.84 EGFR (0.56) EGFRMKNK2MEN1NPC1MAPT
SCHEMBL6996349 0.80 EGFR (0.48) EGFRLMNANPC1RAB9ASMN1; SMN2
SCHEMBL6997797 0.80 EGFR (0.67) EGFRMAPK1HIF1A
SCHEMBL6999229 0.80 EGFR (0.45) EGFRMAPTHPGD
SCHEMBL8487486 0.79 EGFR (0.42) EGFRMEN1NPC1MAPTHPGD
SCHEMBL6997920 0.78 EGFR (0.56) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888351-B1 PYRIMIDO 5,4-D]PYRIMIDINES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION THOMAE GMBH DR K (DE) 2003-10-15 EP disclosed