SCHEMBL6996355

SCHEMBL6996355

CCN1CCN(S(=O)(=O)c2cnc(OCCOC)c(-c3nc4c(-c5ccc(C#N)cc5)n(C)nc4c(=O)[nH]3)c2)CC1

nearest known ligand 0.72

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 20/20 0.72
PDE6C P51160 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994016 0.92 PDE5A (0.76) PDE5APDE6C
SCHEMBL7001475 0.90 PDE5A (0.72) PDE5APDE6C
SCHEMBL7005873 0.90 PDE5A (0.72) PDE5APDE6C
SCHEMBL7001359 0.90 PDE5A (0.73) PDE5APDE6C
SCHEMBL6999125 0.89 PDE5A (0.73) PDE5APDE6C
SCHEMBL7000301 0.89 PDE5A (0.70) PDE5APDE6C
SCHEMBL6999224 0.87 PDE5A (0.73) PDE5APDE6C
SCHEMBL6993435 0.87 PDE5A (0.76) PDE5APDE6C
SCHEMBL7001442 0.86 PDE5A (0.74) PDE5APDE6C
SCHEMBL7001318 0.85 PDE5A (0.81) PDE5APDE6C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1123296-B1 PYRAZOLOPYRIMIDINONE cGMP PDE5 INHIBITORS FOR THE TREATMENT OF SEXUAL DYSFUNCTION PFIZER LTD (GB) 2003-09-17 EP disclosed
US-6333330-B1 Pyrazolopyrimidinone CGMP PDE5 inhibitors for the treatment of sexual dysfunction PFIZER INC. 2001-12-25 US disclosed
EP-1123296-A1 PYRAZOLOPYRIMIDINONE cGMP PDE5 INHIBITORS FOR THE TREATMENT OF SEXUAL DYSFUNCTION Pfizer Limited (GB) 2001-08-16 EP disclosed
WO-2000024745-A1 PYRAZOLOPYRIMIDINONE cGMP PDE5 INHIBITORS FOR THE TREATMENT OF SEXUAL DYSFUNCTION PFIZER LIMITED (GB) 2000-05-04 WO disclosed