SCHEMBL7002888

SCHEMBL7002888

C=CC(=O)Nc1cccc2c(Nc3ccc(Sc4nccn4C)c(Cl)c3)c(C#N)cnc12

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.58
ERBB2 P04626 1/20 0.58
IGF1R P08069 3/20 0.58
MAP2K1 Q02750 17/20 0.57
IKBKB O14920 1/20 0.51
LYN P07948 1/20 0.51
SRC P12931 1/20 0.51
BRAF P15056 1/20 0.51
RPS6KB1 P23443 1/20 0.51
KDR P35968 1/20 0.51
PRKCQ Q04759 1/20 0.51
PDK1 Q15118 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2200467 0.86 IGF1R (0.67) EGFRERBB2IGF1RMAP2K1
SCHEMBL6998144 0.83 IGF1R (0.66) EGFRIGF1RMAP2K1IKBKBLYN
SCHEMBL7000398 0.76 IGF1R (0.75) EGFRERBB2IGF1RMAP2K1
SCHEMBL5255712 0.76 IGF1R (0.68) EGFRERBB2IGF1RMAP2K1
SCHEMBL6381500 0.76 EGFR (0.59) EGFRERBB2
SCHEMBL7002118 0.76 IGF1R (0.74) EGFRERBB2IGF1RMAP2K1
SCHEMBL7001957 0.76 IGF1R (0.71) EGFRERBB2IGF1RMAP2K1
SCHEMBL7001176 0.75 MAP2K1 (0.77) EGFRIGF1RMAP2K1IKBKBLYN
SCHEMBL6381274 0.75 EGFR (0.56) EGFRERBB2PRKCQ
SCHEMBL4894138 0.75 IGF1R (0.68) EGFRIGF1RMAP2K1IKBKBLYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117659-B1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS WYETH CORP (US) 2003-12-03 EP claimed