SCHEMBL7005908

SCHEMBL7005908

CCCCOc1c(CN)n(CC2CC2)c(=O)c2ccc(-c3cnco3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MTOR P42345 1/20 0.39
WNT1 P04628 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
METAP2 P50579 1/20 0.35
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
GPR119 Q8TDV5 2/20 0.34
TLR7 Q9NYK1 5/20 0.33
AAK1 Q2M2I8 2/20 0.33
PIK3CA P42336 1/20 0.33
MMP13 P45452 1/20 0.33
MMP14 P50281 1/20 0.33
DPP4 P27487 2/20 0.33
TLR8 Q9NR97 4/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
HDAC3 O15379 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5235219 0.99 CYP3A4 (0.43) CYP3A4CYP2D6MTORWNT1GSK3B
SCHEMBL5237058 0.87 CYP3A4 (0.40) CYP3A4CYP2D6MTORWNT1GSK3B
Hydrochloric Acid SCHEMBL5234098 0.86 CYP3A4 (0.45) CYP3A4CYP2D6AAK1DPP4
SCHEMBL6110312 0.84 CYP3A4 (0.38) CYP3A4CYP2D6MTORWNT1GSK3B
SCHEMBL5237063 0.83 CYP3A4 (0.40) CYP3A4CYP2D6MTORWNT1GSK3B
SCHEMBL6110309 0.79 CYP3A4 (0.37) CYP3A4CYP2D6MTORWNT1GSK3B
Hydrochloric Acid SCHEMBL5234489 0.78 NPC1 (0.46) DPP4
SCHEMBL27599111 0.78 CYP3A4 (0.46) CYP3A4CYP2D6MTORWNT1GSK3B
Hydrochloric Acid SCHEMBL5231925 0.75 DPP4 (0.51) DPP4
SCHEMBL5236547 0.74 CYP3A4 (0.41) CYP3A4CYP2D6AAK1PIK3CADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed