SCHEMBL700683

SCHEMBL700683

CC1CN(c2ccc(C#N)cc2)CCN1c1nc(-c2ccncc2F)cc(=O)n1C

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.73
CYP2D6 P10635 11/20 0.73
CYP1A2 P05177 8/20 0.61
CYP3A4 P08684 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL696811 1.00 GSK3B (0.73) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL698683 0.91 GSK3B (0.74) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL696862 0.90 GSK3B (0.69) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL696065 0.89 GSK3B (0.64) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL696259 0.89 GSK3B (0.71) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL695999 0.87 GSK3B (0.74) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL695864 0.87 GSK3B (0.79) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL696839 0.87 GSK3B (0.73) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL8234313 0.86 GSK3B (0.61) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL696815 0.86 GSK3B (0.61) GSK3BCYP2D6CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423207-A2 2-(cyclic amino)-pyrimidone derivatives as TPK1 inhibitors Mitsubishi Tanabe Pharma Corporation (JP) 2012-02-29 EP claimed