SCHEMBL7007899

SCHEMBL7007899

CC=C(C)NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 5/20 0.48
KIF11 P52732 1/20 0.36
ALDH1A1 P00352 4/20 0.35
ALOX15 P16050 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 2/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11721973 0.80 KCNN4 (0.50) KCNN4KIF11ALDH1A1ALOX15HDAC3
Hydrochloric Acid SCHEMBL11723541 0.78 KCNN4 (0.48) KCNN4KIF11ALDH1A1ALOX15HDAC3
SCHEMBL8226385 0.76 KCNN4 (0.50) KCNN4KIF11ALDH1A1HDAC3HDAC4
SCHEMBL4078488 0.71 KCNN4 (0.44) KCNN4KIF11ALDH1A1MAPTKMT2A
SCHEMBL316124 0.71 KCNN4 (0.55) KCNN4KIF11ALDH1A1ALOX15HDAC3
SCHEMBL2549817 0.70 KCNN4 (0.54) KCNN4KIF11ALDH1A1ALOX15HDAC3
SCHEMBL10825012 0.70 KCNN4 (0.48) KCNN4KIF11ALDH1A1ALOX15HDAC3
SCHEMBL6906467 0.69 KDM4E (0.55) KCNN4ALDH1A1HDAC3HDAC4HDAC1
SCHEMBL24400266 0.68 KCNN4 (0.52) KCNN4KIF11ALDH1A1HDAC3HDAC4
SCHEMBL28266739 0.68 HDAC3 (0.42) KCNN4ALDH1A1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252162-A4 ALPHA V INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2003-06-11 EP disclosed
EP-1252162-A1 ALPHA V INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2002-10-30 EP disclosed
WO-2001053297-A1 ALPHA V INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2001-07-26 WO disclosed