SCHEMBL7008745

SCHEMBL7008745

CCOC(=O)c1cn(-c2cc(N)c(F)cc2F)c2c(OC)c(F)c(F)cc2c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 3/20 0.52
HTT P42858 1/20 0.43
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 4/20 0.42
HPGD P15428 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HSD17B10 Q99714 2/20 0.42
TOP1 P11387 1/20 0.39
ADRB2 P07550 1/20 0.39
PIM1 P11309 1/20 0.37
IRAK1 P51617 1/20 0.37
CAMK2B Q13554 1/20 0.37
CAMK2G Q13555 1/20 0.37
CAMK2D Q13557 1/20 0.37
PIM3 Q86V86 1/20 0.37
CYP2C19 P33261 1/20 0.37
ROCK2 O75116 1/20 0.36
CDK1 P06493 1/20 0.36
PRKACA P17612 1/20 0.36
CDK2 P24941 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005444 0.91 STAT3 (0.61) STAT3HTTKMT2AKDM4EHPGD
SCHEMBL19729429 0.91 STAT3 (0.49) STAT3HTTKMT2AKDM4EHPGD
SCHEMBL7007194 0.89 STAT3 (0.54) STAT3HTTKMT2AKDM4EHPGD
SCHEMBL7007759 0.87 STAT3 (0.52) STAT3HTTKMT2AKDM4EHPGD
SCHEMBL7009566 0.87 TOP1 (0.52) KMT2AKDM4EHPGDALDH1A1HSD17B10
SCHEMBL9774020 0.85 STAT3 (0.52) STAT3HTTKMT2AKDM4EHPGD
SCHEMBL7005217 0.82 KMT2A (0.56) STAT3HTTKMT2AKDM4EHPGD
SCHEMBL9773968 0.81 HTT (0.54) STAT3HTTKMT2AKDM4EHPGD
SCHEMBL7009131 0.80 STAT3 (0.53) STAT3HTTKMT2AKDM4EHPGD
SCHEMBL1344957 0.80 STAT3 (0.54) STAT3HTTKMT2AKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787720-B1 PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KK (JP) 2003-07-16 EP disclosed
US-5910498-A NOVEL COMPOUNDS HAVING REDUCED CYTOTOXICITY, PHOTOTOXICITY; TREATING BACTERIAL AND VIRAL INFECTIONS WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1999-06-08 US disclosed
EP-0787720-A1 NOVEL PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1997-08-06 EP disclosed