SCHEMBL7012797

SCHEMBL7012797

O[C@@H](COc1ccc(-c2noc3cc(F)ccc23)cc1)CN1CCC(c2ccccc2F)CC1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.58
HTR1A P08908 3/20 0.58
DRD2 P14416 2/20 0.58
TSHR P16473 1/20 0.46
CHRNA7 P36544 1/20 0.45
KCNH2 Q12809 2/20 0.45
HTR7 P34969 2/20 0.45
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5359817 0.90 HTR2A (0.59) HTR2AHTR1ADRD2TSHRCHRNA7
SCHEMBL5364879 0.90 HTR2A (0.59) HTR2AHTR1ADRD2TSHRCHRNA7
SCHEMBL5359826 0.90 HTR2A (0.59) HTR2AHTR1ADRD2TSHRCHRNA7
SCHEMBL5359086 0.88 HTR2A (0.61) HTR2AHTR1ADRD2TSHRUSP2
SCHEMBL5375200 0.88 HTR2A (0.61) HTR2AHTR1ADRD2TSHRUSP2
SCHEMBL5368375 0.88 HTR2A (0.72) HTR2AHTR1ADRD2KCNH2
SCHEMBL5359089 0.88 HTR2A (0.61) HTR2AHTR1ADRD2TSHRUSP2
SCHEMBL5368366 0.88 HTR2A (0.72) HTR2AHTR1ADRD2KCNH2
Hydrochloric Acid SCHEMBL5367657 0.87 HTR2A (0.60) HTR2AHTR1ADRD2TSHR
Hydrochloric Acid SCHEMBL5367650 0.87 HTR2A (0.60) HTR2AHTR1ADRD2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216244-B1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists AVENTIS PHARMA INC (US) 2003-08-13 EP claimed