Ethyne

Ethyne

SCHEMBL7015681

C#C.C[C@@]12CCC[C@H]1[C@@H]1CCC3CCCC[C@@H]3[C@H]1CC2

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 5/20 0.52
GRIN2B Q13224 5/20 0.52
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
NR1I3 Q14994 1/20 0.39
MBOAT4 Q96T53 3/20 0.35
CYP19A1 P11511 3/20 0.33
SHBG P04278 2/20 0.33
AKR1B10 O60218 1/20 0.32
GABRP O00591 2/20 0.31
GABRD O14764 2/20 0.31
GABRA1 P14867 2/20 0.31
GABRB1 P18505 2/20 0.31
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
GABRA5 P31644 2/20 0.31
GABRA3 P34903 2/20 0.31
GABRA2 P47869 2/20 0.31
GABRB2 P47870 2/20 0.31
GABRA4 P48169 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL374356 0.97 GRIN1 (0.55) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL7353210 0.97 GRIN1 (0.55) GRIN1GRIN2BCDK5CDK5R1NR1I3
Charcoal, Activated SCHEMBL4630579 0.95 GRIN1 (0.53) GRIN1GRIN2BCDK5CDK5R1NR1I3
Propane SCHEMBL27462424 0.92 GRIN1 (0.51) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL30645499 0.79 GRIN1 (0.58) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL6853527 0.78 GRIN1 (0.68) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL13007746 0.78 GRIN1 (0.60) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL133513 0.78 GRIN1 (0.60) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL4834976 0.78 GRIN1 (0.56) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL22018389 0.78 GRIN1 (0.60) GRIN1GRIN2BCDK5CDK5R1NR1I3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994713-B1 USE OF A 7alpha-METHYL-17alpha-ETHYNYL-ESTRANE DERIVATIVE FOR THE TREATMENT OF ATHEROSCLEROSIS AKZO NOBEL NV (NL) 2003-11-05 EP disclosed
EP-0994713-A1 USE OF A 7$g(a)-METHYL-17$g(a)-ETHYNYL-ESTRANE DERIVATIVE FOR THE TREATMENT OF ATHEROSCLEROSIS Akzo Nobel N.V. (NL) 2000-04-26 EP disclosed