SCHEMBL7021941

SCHEMBL7021941

C[C@H](Nc1nccc(-n2cnc3cc(NC(=O)c4ccco4)ccc32)n1)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LCK P06239 11/20 0.64
NPC1 O15118 7/20 0.62
RAB9A P51151 7/20 0.62
SMN1; SMN2 Q16637 4/20 0.62
TP53 P04637 3/20 0.62
ALDH1A1 P00352 1/20 0.62
HPGD P15428 1/20 0.62
HSD17B10 Q99714 1/20 0.62
JAK2 O60674 1/20 0.55
JAK3 P52333 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020233 0.94 LCK (0.63) LCKNPC1RAB9ASMN1; SMN2TP53
SCHEMBL7014887 0.89 LCK (0.69) LCKNPC1RAB9AJAK2JAK3
SCHEMBL7016999 0.88 LCK (0.63) LCKALDH1A1JAK2JAK3
SCHEMBL7024707 0.88 LCK (0.71) LCKNPC1RAB9AJAK2JAK3
SCHEMBL7021308 0.87 LCK (0.65) LCKNPC1RAB9ASMN1; SMN2JAK2
SCHEMBL7017985 0.87 LCK (0.67) LCKNPC1RAB9AJAK2JAK3
SCHEMBL7017212 0.87 LCK (0.69) LCKNPC1RAB9AJAK2JAK3
SCHEMBL7588436 0.87 LCK (0.69) LCKNPC1RAB9AJAK2JAK3
SCHEMBL7022787 0.86 LCK (0.70) LCKNPC1RAB9AJAK2JAK3
SCHEMBL7017343 0.86 LCK (0.68) LCKJAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206265-B1 SRC KINASE INHIBITOR COMPOUNDS MERCK & CO INC (US) 2003-11-12 EP disclosed
US-6498165-B1 PYRIMIDINE COMPOUNDS; PROPHYLAXIS AND TREATMENT OF SUCH AS IMMUNE DISEASES, HYPERPROLIFERATIVE DISORDERS, CANCER, ANGIOGENSIS, ATHEROSCELEROSIS, GRAFT REJECTION, RHEUMATOID ARTHRITIS, PSORIASIS MERCK & CO., INC. 2002-12-24 US disclosed