SCHEMBL7025484

SCHEMBL7025484

N[C@@](O)(C(=O)O)[C@@H](O)[C@H](O)[C@@H](O)CO

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.47
SLCO1B1 Q9Y6L6 1/20 0.47
PDE4A P27815 1/20 0.45
LMNA P02545 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TDP1 Q9NUW8 1/20 0.40
OR51E2 Q9H255 1/20 0.32
KDM4E B2RXH2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28449969 1.00 USP2 (0.47) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL8356023 1.00 USP2 (0.47) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL17888974 0.94 USP2 (0.50) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL5960037 0.83 USP2 (0.42) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL9392459 0.83 USP2 (0.42) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL28240342 0.83 USP2 (0.42) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL8413989 0.81 USP2 (0.41) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL8497603 0.80 USP2 (0.41) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL9763747 0.80 USP2 (0.48) USP2SLCO1B1PDE4ALMNAL3MBTL1
SCHEMBL18825609 0.80 USP2 (0.48) USP2SLCO1B1PDE4ALMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939831-B1 NOVEL BACTERIAL STRAINS AND USE THEREOF IN FERMENTATION PROCESSES FOR 2-KETO-L-GULONIC ACID PRODUCTION ARCHER DANIELS MIDLAND CO (US) 2003-07-09 EP disclosed
US-6541239-B1 From L-sorbose, using pure culture of microorganisms which has been transformed with linear or circular DNA ARCHER-DANIELS-MIDLAND COMPANY 2003-04-01 US disclosed
EP-1278879-A1 BACTERIAL STRAINS AND FERMENTATION PROCESSES FOR THE PRODUCTION OF 2-KETO-L-GULONIC ACID Archer-Daniels-Midland Company (US) 2003-01-29 EP disclosed
US-6387654-B1 FOR SIMPLE, SHORTER AND EFFICIENT PRODUCTION FROM D-SORBITOL VIA L-SORBOSE IN MIXED CULTURE ARCHER-DANIELS-MIDLAND COMPANY 2002-05-14 US disclosed
US-6319699-B1 GENERATING PREFERENTIAL COMPOUNDS IN CULTURE; TRANSFORM MMICROORGANISM, CULTURE IN SORBOSE AND CULTURE BROTH, RECOVER PREFERENTIAL COMPOUNDS ARCHER-DANIELS-MIDLAND COMPANY 2001-11-20 US disclosed
WO-2001083798-A1 BACTERIAL STRAINS AND FERMENTATION PROCESSES FOR THE PRODUCTION OF 2-KETO-L-GULONIC ACID ARCHER-DANIELS-MIDLAND COMPANY (US) 2001-11-08 WO disclosed
CN-1246156-A Novel bacterial strains and use thereof in fermentation processes for 2-keto-L-gulonic acid production ARCHER DANIELS MIDLAND CO (US) 2000-03-01 CN disclosed
US-5989891-A SELECTIVELY CULTURING FOR MICROORGANISMAL CELLS CAPABLE OF GROWTH IN PRESENCE OF INHIBITING AMOUNTS OF 2-KETO-L-GULONIC ACID DERIVATIVE OR ANALOG; FOR EFFICIENT PRODUCTION ARCHER-DANIELS-MIDLAND COMPANY (US) 1999-11-23 US disclosed
EP-0939831-A1 NOVEL BACTERIAL STRAINS AND USE THEREOF IN FERMENTATION PROCESSES FOR 2-KETO-L-GULONIC ACID PRODUCTION ARCHER-DANIELS-MIDLAND COMPANY (US) 1999-09-08 EP disclosed
US-5834231-A FERMENTATIVE CONVERSION OF L-SORBOSE AND/OR D-SORBITOL ARCHER DANIELS MIDLAND CO. (US) 1998-11-10 US disclosed
WO-1998017819-A1 NOVEL BACTERIAL STRAINS AND USE THEREOF IN FERMENTATION PROCESSES FOR 2-KETO-L-GULONIC ACID PRODUCTION ARCHER-DANIELS-MIDLAND COMPANY (US) 1998-04-30 WO disclosed