SCHEMBL7028796

SCHEMBL7028796

C#Cc1cccc(Nc2ncnc3[nH]cc(OC(=O)OC)c23)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.51
GAK O14976 3/20 0.51
FBP1 P09467 2/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.51
AURKA O14965 2/20 0.49
RPS6KB1 P23443 1/20 0.49
DYRK1A Q13627 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
ERBB2 P04626 5/20 0.47
RIPK2 O43353 2/20 0.47
BUB1 O43683 2/20 0.47
STK10 O94804 2/20 0.47
ABL1 P00519 2/20 0.47
LCK P06239 2/20 0.47
LYN P07948 2/20 0.47
RET P07949 2/20 0.47
SRC P12931 2/20 0.47
FGFR2 P21802 2/20 0.47
FECH P22830 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7020994 0.99 EGFR (0.50) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7021138 0.84 AURKA (0.53) EGFRGAKFBP1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL7021133 0.83 AURKA (0.53) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7025011 0.80 AURKA (0.56) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7022596 0.80 BRAF (0.60) EGFRGAKFBP1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL7017702 0.79 BRAF (0.59) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7016150 0.78 BRAF (0.58) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7024764 0.78 AURKA (0.49) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7019299 0.77 EGFR (0.51) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL3535063 0.77 BRAF (0.59) EGFRGAKFBP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0831829-B1 HETEROCYCLIC RING-FUSED PYRIMIDINE DERIVATIVES PFIZER (US) 2003-08-20 EP claimed