SCHEMBL7029374

SCHEMBL7029374

O=c1[nH]c(=O)c2c(Cl)c(Br)ccc2[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.38
CA9 Q16790 2/20 0.38
KDM4E B2RXH2 1/20 0.38
PARP1 P09874 1/20 0.38
TYMP P19971 5/20 0.36
GRIA1 P42261 2/20 0.35
CACNG8 Q8WXS5 2/20 0.35
ALDH1A1 P00352 5/20 0.35
MAPT P10636 5/20 0.35
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
PAX8 Q06710 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7032754 0.82 CA12 (0.39) CA12CA9KDM4EPARP1TYMP
SCHEMBL7027462 0.82 GRIN2D (0.50) CA12CA9KDM4EPARP1TYMP
SCHEMBL31621485 0.79 PTK6 (0.38) CA12CA9KDM4EPARP1TYMP
SCHEMBL7032399 0.79 GRIA1 (0.38) CA12CA9KDM4EPARP1TYMP
SCHEMBL24815911 0.79 DAO (0.46) CA12CA9KDM4EPARP1TYMP
SCHEMBL18554548 0.78 IDH1 (0.38) CA12CA9KDM4EPARP1GRIA1
SCHEMBL30013511 0.74 FEN1 (0.50) CA12CA9KDM4EPARP1TYMP
SCHEMBL1502649 0.74 FEN1 (0.50) CA12CA9KDM4EPARP1TYMP
SCHEMBL4707223 0.74 CA12 (0.46) CA12CA9GRIA1ALDH1A1MAPT
SCHEMBL29204414 0.73 PARP1 (0.48) CA12CA9KDM4EPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed