SCHEMBL7030828

SCHEMBL7030828

O=c1[nH]c(=O)c2cccc(OC(F)(F)F)c2[nH]1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.58
GRIA1 P42261 2/20 0.43
CACNG8 Q8WXS5 2/20 0.43
TRPA1 O75762 1/20 0.41
CA12 O43570 1/20 0.41
PARP1 P09874 1/20 0.41
CA9 Q16790 1/20 0.41
BRAF P15056 8/20 0.40
PGR P06401 1/20 0.36
C1R P00736 1/20 0.36
POLB P06746 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
NQO2 P16083 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HCAR1 Q9BXC0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7029217 0.84 KDM4E (0.41) KDM4ECA12PARP1CA9POLB
SCHEMBL3423322 0.78 NQO2 (0.57) KDM4EPARP1POLBTNKSTNKS2
SCHEMBL20954833 0.75 KDM4E (0.57) KDM4ECA12PARP1CA9POLB
SCHEMBL7033735 0.74 KDM4E (0.41) KDM4ECA12PARP1CA9POLB
SCHEMBL7027327 0.74 KDM4E (0.41) KDM4ECA12PARP1CA9POLB
SCHEMBL7030040 0.74 KDM4E (0.41) KDM4ECA12PARP1CA9POLB
SCHEMBL7032421 0.74 KDM4E (0.41) KDM4ECA12PARP1CA9POLB
SCHEMBL7030573 0.74 DAO (0.49) KDM4ECA12PARP1CA9POLB
SCHEMBL7031280 0.74 PARP1 (0.41) KDM4ECA12PARP1CA9POLB
SCHEMBL8496530 0.74 GRIA1 (0.49) KDM4EGRIA1CACNG8CA12PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed