SCHEMBL703142

SCHEMBL703142

Cn1nc(CNC2CN3CCC2CC3)c2c(C(=O)O)cccc21.[LiH]

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.41
ADRA2A P08913 2/20 0.41
CHRM1 P11229 2/20 0.41
ADRA2B P18089 2/20 0.41
CHRM3 P20309 2/20 0.41
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR4 Q13639 2/20 0.41
CYP1A2 P05177 1/20 0.41
CHRM4 P08173 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
ALOX15 P16050 1/20 0.41
HTR1D P28221 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
GAA P10253 1/20 0.39
HTR3A P46098 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4316908 0.99 CHRM2 (0.41) CHRM2ADRA2ACHRM1ADRA2BCHRM3
SCHEMBL700319 0.99 CHRM2 (0.41) CHRM2ADRA2ACHRM1ADRA2BCHRM3
SCHEMBL4317776 0.99 CHRM2 (0.41) CHRM2ADRA2ACHRM1ADRA2BCHRM3
SCHEMBL700432 0.90 CHRM2 (0.40) CHRM2ADRA2ACHRM1ADRA2BCHRM3
SCHEMBL4314155 0.89 CHRM2 (0.40) CHRM2ADRA2ACHRM1ADRA2BCHRM3
SCHEMBL4314161 0.89 CHRM2 (0.40) CHRM2ADRA2ACHRM1ADRA2BCHRM3
SCHEMBL701021 0.89 CHRM2 (0.42) CHRM2ADRA2ACHRM1ADRA2BCHRM3
SCHEMBL700878 0.89 CHRM2 (0.42) CHRM2ADRA2ACHRM1ADRA2BCHRM3
Lithium Ion SCHEMBL701319 0.89 CHRM2 (0.40) CHRM2ADRA2ACHRM1ADRA2BCHRM3
Lithium Ion SCHEMBL701018 0.89 CHRM2 (0.40) CHRM2ADRA2ACHRM1ADRA2BCHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8124600-B2 5-HT3 receptor modulators, methods of making, and use thereof ALBANY MOLECULAR RESEARCH, INC. (US) 2012-02-28 US disclosed