SCHEMBL7032724

SCHEMBL7032724

CNC(=O)C(N)Cc1cc(Cl)ccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 16/20 0.50
ALDH1A1 P00352 1/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC3 O15379 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7032727 1.00 HDAC8 (0.50) HDAC8ALDH1A1HDAC1HDAC3HDAC2
SCHEMBL7032203 0.88 HDAC8 (0.63) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL7032205 0.88 HDAC8 (0.63) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL29398382 0.81 CYP2C9 (0.51) HDAC8ALDH1A1HDAC1HDAC3HDAC2
SCHEMBL21690291 0.81 CYP2C9 (0.51) HDAC8ALDH1A1HDAC1HDAC3HDAC2
SCHEMBL29398451 0.81 CYP2C9 (0.51) HDAC8ALDH1A1HDAC1HDAC3HDAC2
Hydrochloric Acid SCHEMBL27557729 0.81 HDAC8 (0.46) HDAC8ALDH1A1HDAC1HDAC3HDAC2
SCHEMBL7033985 0.78 CTSC (0.52)
SCHEMBL7033988 0.78 CTSC (0.52)
Hydrochloric Acid SCHEMBL27578024 0.77 CYP3A4 (0.45) HDAC8ALDH1A1HDAC1HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0977730-B1 AMINO ACID DERIVATIVES INHIBITING EXTRACELLULAR MATRIX METALLOPROTEINASE AND TNF ALPHA RELEASE CHIESI FARMA SPA (IT) 2003-03-12 EP disclosed
EP-0977730-A1 AMINO ACID DERIVATIVES INHIBITING EXTRACELLULAR MATRIX METALLOPROTEINASE AND TNF ALPHA RELEASE CHIESI FARMACEUTICI S.p.A. (IT) 2000-02-09 EP disclosed
WO-1998047863-A1 AMINO ACID DERIVATIVES INHIBITING EXTRACELLULAR MATRIX METALLOPROTEINASE AND TNF ALPHA RELEASE CHIESI FARMACEUTICI S.P.A. (IT) 1998-10-29 WO disclosed