SCHEMBL7033757

SCHEMBL7033757

CC/C=C/c1ccc2c(=O)[nH]c(=O)[nH]c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMP P19971 3/20 0.43
PARP1 P09874 3/20 0.42
KDM4E B2RXH2 2/20 0.42
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
P2RY12 Q9H244 2/20 0.34
GSK3B P49841 1/20 0.34
KIF11 P52732 1/20 0.34
IP6K1 Q92551 1/20 0.34
PDE3B Q13370 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7033759 1.00 TYMP (0.43) TYMPPARP1KDM4ECA12CA9
SCHEMBL7027670 0.88 TYMP (0.46) TYMPPARP1KDM4ECA12CA9
SCHEMBL7027667 0.88 TYMP (0.46) TYMPPARP1KDM4ECA12CA9
SCHEMBL7030723 0.88 CA12 (0.44) TYMPPARP1KDM4ECA12CA9
SCHEMBL7030725 0.88 CA12 (0.44) TYMPPARP1KDM4ECA12CA9
SCHEMBL7024197 0.85 PARP1 (0.42) TYMPPARP1KDM4ECA12CA9
SCHEMBL7024202 0.85 PARP1 (0.42) TYMPPARP1KDM4ECA12CA9
SCHEMBL7022550 0.83 PARP1 (0.46) TYMPPARP1KDM4ECA12CA9
SCHEMBL7022549 0.83 PARP1 (0.46) TYMPPARP1KDM4ECA12CA9
SCHEMBL3380424 0.78 KDM4E (0.53) PARP1KDM4ECA12CA9KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed