SCHEMBL7038181

SCHEMBL7038181

CN(CCC[C@H](C(N)=O)N(Cc1ccc(O)cc1)C(=O)C(c1ccccc1)c1ccccc1)C(=N)N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
TACR1 P25103 3/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
NPY1R P25929 2/20 0.39
KDM4E B2RXH2 2/20 0.37
ATM Q13315 1/20 0.37
MTOR P42345 1/20 0.37
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
GLI1 P08151 1/20 0.35
GLI2 P10070 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
NPFFR1 Q9GZQ6 1/20 0.34
NPFFR2 Q9Y5X5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4702218 0.99 TDP1 (0.42) TDP1MEN1KMT2ATACR1NOS3
SCHEMBL8112100 0.90 TDP1 (0.44) TDP1MEN1KMT2ATACR1NPY1R
SCHEMBL7043265 0.88 TDP1 (0.42) TDP1MEN1KMT2A
SCHEMBL8612230 0.88 TDP1 (0.42) TDP1MEN1KMT2A
SCHEMBL1389094 0.85 TDP1 (0.38) TDP1MEN1KMT2ANPY1RNPFFR1
SCHEMBL7750469 0.85 TDP1 (0.38) TDP1MEN1KMT2ANPY1RNPFFR1
SCHEMBL8126608 0.84 TDP1 (0.41) TDP1MEN1KMT2ANPY1RNPFFR1
Hydrochloric Acid SCHEMBL8120018 0.84 TDP1 (0.37) TDP1MEN1KMT2ANPY1RNPFFR1
SCHEMBL8119409 0.83 EPOR (0.43) TDP1MEN1KMT2ANPY1RNPFFR1
SCHEMBL1593414 0.83 NPY1R (0.42) TDP1NPY1RNPFFR1NPFFR2NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-B1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM THOMAE GMBH DR K (DE) 2003-03-26 EP claimed
EP-0885186-B1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM THOMAE GMBH DR K (DE) 2003-03-26 EP disclosed