SCHEMBL70399

SCHEMBL70399

Nc1cncc(F)c1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30644320 1.00
Hydrochloric Acid SCHEMBL4605896 0.97 HCAR2 (0.41)
Hydrochloric Acid SCHEMBL3934248 0.97
Formaldehyde SCHEMBL29107865 0.93 HCAR2 (0.43)
SCHEMBL56635 0.78
SCHEMBL187404 0.78
Bromide SCHEMBL7898147 0.76 MEN1 (0.50)
Hydrochloric Acid SCHEMBL3583511 0.76
Ammonia Solution, Strong SCHEMBL28242958 0.76 HCAR2 (0.50)
SCHEMBL21044202 0.72 TAAR1 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 774 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260098018-A1 BICYCLIC 1,4-DIAZEPANONES AND THERAPEUTIC USES THEREOF CYTOKINETICS INC (US) 2026-04-09 US claimed
US-12479824-B2 Method for preparing ivosidenib and an intermediate thereof SERVIER PHARMACEUTICALS LLC (US) 2025-11-25 US claimed
CN-119899194-B Bicyclic heteroaryl BRAF negative allosteric modulator, and preparation method and application thereof 浙江省人民医院 2025-06-24 CN claimed
CN-119899194-A Bicyclic heteroaryl BRAF negative allosteric modulator, and preparation method and application thereof 浙江省人民医院 2025-04-29 CN claimed
CN-119432148-A Perovskite ink, perovskite film and battery device 云南大学 2025-02-14 CN claimed
CN-119082658-A High-strength and high-toughness microalloy structural steel and preparation method thereof 河北纵横集团丰南钢铁有限公司 2024-12-06 CN claimed
CN-114555584-B Ai Funi cloth (IVOSIDENIB) and process for producing intermediate thereof 法国施维雅药厂 2024-07-05 CN claimed
EP-4010331-B1 A METHOD FOR PREPARING IVOSIDENIB AND AN INTERMEDIATE THEREOF SERVIER LAB (FR) 2023-10-04 EP claimed
US-20230025411-A1 A METHOD FOR PREPARING IVOSIDENIB AND AN INTERMEDIATE THEREOF SERVIER PHARMACEUTICALS LLC 2023-01-26 US claimed
EP-4010331-A1 A METHOD FOR PREPARING IVOSIDENIB AND AN INTERMEDIATE THEREOF Les Laboratoires Servier (FR) 2022-06-15 EP claimed
WO-2021079380-A1 IMPROVED PROCESS FOR THE PREPARATION OF (2S)-N-{(1S)-1-(2-CHLOROPHENYL)-2-[(3,3-DIFLUOROCYCLOBUTYL)-AMINO]-2-OXOETHYL}-1-(4-CYANOPYRIDIN-2-YL)-N-(5-FLUOROPYRIDIN-3-YL)-5-OXOPYRROLIDINE-2-CARBOXAMIDE MSN LABORATORIES PRIVATE LIMITED, R&D CENTER (IN) 2021-04-29 WO claimed
CN-112367995-A Evonib forms and pharmaceutical compositions 安吉奥斯医药品有限公司 2021-02-12 CN claimed
WO-2021026436-A1 A METHOD FOR PREPARING IVOSIDENIB AND AN INTERMEDIATE THEREOF AGIOS PHARMACEUTICALS, INC. (US) 2021-02-11 WO claimed
CN-111349081-B Chiral synthesis method of Ivosidenib and intermediate thereof 宁波大学科学技术学院 2021-01-15 CN claimed
CN-109678793-B Preparation method of 5-fluoro-3-aminopyridine 上海卡洛化学有限公司 2020-08-04 CN claimed
CN-111349081-A Chiral synthesis method of Ivosidenib and intermediate thereof 宁波大学科学技术学院 2020-06-30 CN claimed
US-20150274661-A1 INDOL-AMIDE COMPOUNDS AS BETA-AMYLOID INHBITORS HOFFMANN-LA ROCHE INC. (US) 2015-10-01 US claimed
EP-2909190-A1 INDOL-AMIDE COMPOUNDS AS BETA-AMYLOID INHBITORS F. Hoffmann-La Roche AG (CH) 2015-08-26 EP claimed
WO-2014060386-A1 INDOL-AMIDE COMPOUNDS AS BETA-AMYLOID INHBITORS F. HOFFMANN-LA ROCHE AG (CH) 2014-04-24 WO claimed
EP-2722329-A1 Indol-amide compounds as beta-amyloid inhbitors F. Hoffmann-La Roche AG (CH) 2014-04-23 EP claimed