SCHEMBL7042142

SCHEMBL7042142

CCCN1CCC(c2nc3c(OC(N)=O)cccc3n2CCN2CCCCC2)C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.52
PARP2 Q9UGN5 1/20 0.42
CYP2D6 P10635 2/20 0.39
HPGD P15428 2/20 0.39
MEN1 O00255 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
PKM P14618 1/20 0.39
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39
KDM2B Q8NHM5 1/20 0.39
HRH1 P35367 3/20 0.38
DRD3 P35462 1/20 0.38
DRD2 P14416 1/20 0.38
KCNH2 Q12809 1/20 0.38
ACHE P22303 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7043782 0.99 PARP1 (0.52) PARP1PARP2CYP2D6MEN1CYP3A4
SCHEMBL7043532 0.97 PARP1 (0.48) PARP1PARP2CYP2D6KDM2BHRH1
SCHEMBL7043437 0.96 PARP1 (0.49) PARP1PARP2CYP2D6KDM2BHRH1
SCHEMBL7042613 0.96 PARP1 (0.56) PARP1PARP2CYP2D6HPGDMEN1
SCHEMBL7046731 0.95 PARP1 (0.56) PARP1PARP2CYP2D6HPGDMEN1
SCHEMBL7035297 0.90 PARP1 (0.52) PARP1PARP2KDM2BHRH1DRD3
SCHEMBL7042319 0.90 PARP1 (0.52) PARP1PARP2CYP2D6KDM2BHRH1
SCHEMBL7044350 0.90 PARP1 (0.53) PARP1PARP2KDM2BHRH1DRD3
SCHEMBL7042194 0.89 PARP1 (0.47) PARP1CYP2D6KDM2BHRH1DRD3
SCHEMBL7045127 0.89 PARP1 (0.47) PARP1CYP2D6KDM2BHRH1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed