SCHEMBL7043404

SCHEMBL7043404

CCCc1c(OCCCNc2ccc(C(C)C(=O)O)cc2Cl)ccc2c(CC(C)(C)C)noc12

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 16/20 0.46
PPARG P37231 16/20 0.46
PPARA Q07869 14/20 0.46
NR1H2 P55055 7/20 0.46
NR1H3 Q13133 7/20 0.46
GRM2 Q14416 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7039181 0.86 PPARD (0.62) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL8668801 0.84 GRM2 (0.50) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL7044849 0.84 PPARD (0.54) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL7044850 0.78 PPARA (0.69) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL7039142 0.78 PPARA (0.75) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL6368217 0.76 GRM2 (0.59) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL5953747 0.75 GRM2 (0.59) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL6367383 0.74 GRM2 (0.55) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL7043426 0.74 PPARA (0.60) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL5954097 0.74 GRM2 (0.56) PPARDPPARGPPARANR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882029-B1 HETEROCYCLIC DERIVATIVES AS ANTIDIABETIC AND ANTIOBESITY AGENTS MERCK & CO INC (US) 2003-04-02 EP claimed