SCHEMBL7047730

SCHEMBL7047730

[CH2]NC(=O)C1OC1C(=O)OCC

nearest known ligand 0.73

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 6/20 0.48
CTSL P07711 3/20 0.48
CTSB P07858 2/20 0.48
LMNA P02545 1/20 0.48
CTSG P08311 1/20 0.48
TSHR P16473 1/20 0.45
PPM1B O75688 1/20 0.39
PTPN1 P18031 1/20 0.39
PPP1CC P36873 1/20 0.39
MGAM O43451 1/20 0.37
GAA P10253 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
ALDH1A1 P00352 2/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2387693 0.85 TSHR (0.55) CAPN1CTSLCTSBLMNACTSG
SCHEMBL5317413 0.85 TSHR (0.55) CAPN1CTSLCTSBLMNACTSG
SCHEMBL2387697 0.85 TSHR (0.55) CAPN1CTSLCTSBLMNACTSG
SCHEMBL11545787 0.85 TSHR (0.55) CAPN1CTSLCTSBLMNACTSG
SCHEMBL2387688 0.85 TSHR (0.55) CAPN1CTSLCTSBLMNACTSG
SCHEMBL7047733 0.85 CAPN1 (0.48) CAPN1CTSLCTSBLMNACTSG
SCHEMBL5556039 0.83 TSHR (0.53) CAPN1CTSLCTSBLMNACTSG
SCHEMBL15171333 0.80 CAPN1 (0.58) CAPN1CTSLCTSBLMNACTSG
SCHEMBL14067709 0.80 CAPN1 (0.51) CAPN1CTSLCTSBLMNACTSG
SCHEMBL11171419 0.80 CAPN1 (0.51) CAPN1CTSLCTSBLMNACTSG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1029869-B1 Endothelin converting enzyme inhibitors WELLCOME FOUND (GB) 2003-04-23 EP disclosed
US-6235717-B1 Pharmaceutical compounds GLAXO WELLCOME INC. 2001-05-22 US disclosed
EP-1029869-A1 Endothelin converting enzyme inhibitors THE WELLCOME FOUNDATION LIMITED (GB) 2000-08-23 EP disclosed
EP-0677059-A1 ENDOTHELIN CONVERTING ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-10-18 EP disclosed
WO-1994015956-A1 ENDOTHELIN CONVERTING ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-07-21 WO disclosed