SCHEMBL7048275

SCHEMBL7048275

O=C1Nc2ccc(Cl)c(Cl)c2C(=O)C1=NO

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CES1 P23141 9/20 0.67
GALR3 O60755 2/20 0.38
TGM2 P21980 3/20 0.34
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
LRRK2 Q5S007 2/20 0.32
PDE7A Q13946 1/20 0.32
IDO1 P14902 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7048273 1.00 CES1 (0.67) CES1GALR3TGM2HTR2AHTR2C
SCHEMBL6322718 0.90 CES1 (0.61) CES1GALR3TGM2HTR2AHTR2C
SCHEMBL6316168 0.90 CES1 (0.61) CES1GALR3TGM2HTR2AHTR2C
SCHEMBL7054756 0.81 CES1 (0.46) CES1GALR3TGM2
SCHEMBL7054760 0.81 CES1 (0.46) CES1GALR3TGM2
SCHEMBL734955 0.81 CES1 (1.00) CES1TGM2PDE7A
SCHEMBL7050698 0.81 CES1 (0.42) CES1GALR3TGM2CA1CA2
SCHEMBL7050694 0.81 CES1 (0.42) CES1GALR3TGM2CA1CA2
SCHEMBL5752424 0.77 CES1 (0.61) CES1GALR3TGM2HTR2AHTR2C
SCHEMBL8872679 0.76 CES1 (0.41) CES1GALR3TGM2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5652368-A NERVOUS SYSTEM DISORDERS, ALZHEIMER'S DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-07-29 US disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed