SCHEMBL7050413

SCHEMBL7050413

CCOC(=NNc1ccccc1)C(=O)C(=O)C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 8/20 0.49
LMNA P02545 3/20 0.49
ALDH1A1 P00352 5/20 0.48
NPSR1 Q6W5P4 2/20 0.48
HPGD P15428 1/20 0.48
ATM Q13315 1/20 0.48
MAPT P10636 6/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
KMT2A Q03164 5/20 0.41
MEN1 O00255 3/20 0.41
RECQL P46063 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
CES2 O00748 1/20 0.40
ACHE P22303 1/20 0.40
CES1 P23141 1/20 0.40
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
KYAT1 Q16773 1/20 0.39
ALOX12 P18054 1/20 0.39
MAPK1 P28482 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7046248 0.83 GAA (0.57) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL7050416 0.81 GAA (0.55) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL7484968 0.81 GAA (0.55) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL7041161 0.76 GAA (0.52) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL5253476 0.71 GAA (0.63) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL10141247 0.71 GAA (0.63) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL5253472 0.71 GAA (0.63) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL13901608 0.71 GAA (0.63) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL11753054 0.71 GAA (0.63) GAALMNAALDH1A1NPSR1HPGD
SCHEMBL13664158 0.70 GAA (0.62) GAALMNAALDH1A1NPSR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054667-B1 BICYCLIC PYRROLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIINFLAMMATORY AND IMMUNOMODULATING AGENTS ASTRAZENECA UK LTD (GB) 2003-04-16 EP disclosed
US-6291507-B1 INHIBITOR OF MONOCYTE CHEMOATTRACTANT PROTEIN-1; INDOLE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 2001-09-18 US disclosed