SCHEMBL7053705

SCHEMBL7053705

O=C1Nc2cc(C(F)(F)F)cc(Cl)c2C(=O)/C1=N/O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 5/20 0.44
GALR3 O60755 1/20 0.35
JUN P05412 4/20 0.33
NFKB1 P19838 4/20 0.33
NFKB2 Q00653 4/20 0.33
RELA Q04206 4/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
RECQL P46063 1/20 0.33
PBRM1 Q86U86 1/20 0.32
KDR P35968 1/20 0.31
STK10 O94804 1/20 0.30
SLK Q9H2G2 1/20 0.30
DNMT1 P26358 1/20 0.30
ACE2 Q9BYF1 1/20 0.30
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7053708 1.00 CES1 (0.44) CES1GALR3JUNNFKB1NFKB2
SCHEMBL8871331 0.90 CES1 (0.45) CES1GALR3JUNNFKB1NFKB2
SCHEMBL8871333 0.90 CES1 (0.45) CES1GALR3JUNNFKB1NFKB2
SCHEMBL7054973 0.84 GALR3 (0.36) GALR3JUNNFKB1NFKB2RELA
SCHEMBL7054970 0.84 GALR3 (0.36) GALR3JUNNFKB1NFKB2RELA
SCHEMBL7052798 0.83 GALR3 (0.35) GALR3KDRACE2
SCHEMBL7052801 0.83 GALR3 (0.35) GALR3KDRACE2
SCHEMBL7052297 0.82 CES1 (0.66) CES1DNMT1
SCHEMBL8874088 0.82 CES1 (0.66) CES1DNMT1
SCHEMBL7052301 0.82 CES1 (0.66) CES1DNMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5652368-A NERVOUS SYSTEM DISORDERS, ALZHEIMER'S DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-07-29 US disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed