SCHEMBL7054403

SCHEMBL7054403

N#Cc1ccccc1Oc1ccccc1C#N

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.64
POLB P06746 1/20 0.64
TSHR P16473 2/20 0.48
MAP4K4 O95819 1/20 0.45
AR P10275 1/20 0.44
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
MAPK14 Q16539 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GCK P35557 1/20 0.43
PIN1 Q13526 1/20 0.43
MAPK1 P28482 1/20 0.42
IMPDH2 P12268 1/20 0.42
IMPDH1 P20839 1/20 0.42
LRRK2 Q5S007 1/20 0.42
SLC22A12 Q96S37 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8431375 0.97 GAA (0.62) GAAPOLBTSHRMAP4K4AR
SCHEMBL11115045 0.87 GAA (0.53) GAAPOLBTSHRMAP4K4AR
SCHEMBL18603934 0.87 POLB (0.53) GAAPOLBTSHRMAP4K4AR
SCHEMBL9131619 0.87 GAA (0.53) GAAPOLBTSHRMAP4K4AR
SCHEMBL7807009 0.87 GAA (0.53) GAAPOLBTSHRMAP4K4AR
SCHEMBL30872202 0.87 POLB (0.53) GAAPOLBTSHRMAP4K4AR
SCHEMBL3384331 0.87 GAA (0.53) GAAPOLBTSHRMAP4K4AR
SCHEMBL28625665 0.87 AR (0.61) GAAPOLBTSHRARSMN1; SMN2
SCHEMBL1162713 0.86 GAA (0.72) GAAPOLBTSHRARPDE4A
SCHEMBL30441601 0.86 GAA (0.72) GAAPOLBTSHRARPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104710387-A Disulfonamide macrocyclic compound and synthesis method thereof UNIV SOUTH CHINA NORMAL 2015-06-17 CN claimed
JP-6279389-A None JP disclosed
US-20170073460-A1 POLYETHER KETONE COMPOUND AJINOMOTO CO., INC. (JP) 2017-03-16 US disclosed
CN-104710387-A Disulfonamide macrocyclic compound and synthesis method thereof UNIV SOUTH CHINA NORMAL 2015-06-17 CN disclosed
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed
JP-H06279389-A AMIDINOPHENYL ETHER DERIVATIVE TERUMO CORP 1994-10-04 JP disclosed
US-5084085-A Plant growth regulators FMC CORPORATION (US) 1992-01-28 US disclosed