Bromide

Bromide

SCHEMBL7055840

Br.Cc1ccc(-c2ccccn2)cc1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
PKM P14618 2/20 0.57
KDM4E B2RXH2 6/20 0.54
LMNA P02545 3/20 0.54
CYP1A2 P05177 2/20 0.54
CCR1 P32246 2/20 0.54
CCR5 P51681 2/20 0.54
CCR8 P51685 2/20 0.54
POLB P06746 1/20 0.54
METAP1 P53582 1/20 0.54
BLM P54132 1/20 0.54
HIF1A Q16665 1/20 0.54
DOHH Q9BU89 1/20 0.54
P4HTM Q9NXG6 1/20 0.54
CYP2D6 P10635 1/20 0.53
CYP19A1 P11511 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29577473 0.98 TP53 (0.59) TP53MEN1KMT2APKMKDM4E
SCHEMBL39128 0.98 TP53 (0.59) TP53MEN1KMT2APKMKDM4E
SCHEMBL12339129 0.96 TP53 (0.57) TP53MEN1KMT2APKMKDM4E
SCHEMBL17709417 0.96 TP53 (0.57) TP53MEN1KMT2APKMKDM4E
SCHEMBL17709414 0.96 TP53 (0.57) TP53MEN1KMT2APKMKDM4E
SCHEMBL1815589 0.96 TP53 (0.57) TP53MEN1KMT2APKMKDM4E
Hydrochloric Acid SCHEMBL7060038 0.96 TP53 (0.57) TP53MEN1KMT2APKMKDM4E
SCHEMBL17709412 0.96 TP53 (0.57) TP53MEN1KMT2APKMKDM4E
SCHEMBL17709413 0.96 TP53 (0.57) TP53MEN1KMT2APKMKDM4E
SCHEMBL346638 0.96 TP53 (0.57) TP53MEN1KMT2APKMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979820-B1 2-Phenylpyridine derivatives and production method thereof SUMIKA FINE CHEMICALS CO LTD (JP) 2003-05-07 EP disclosed
US-6268503-B1 REACTING 2-(4-BROMOMETHYLPHENYL)PYRIDINE SALT OR 2-(4-DIBROMOMETHYLPHENYL)PYRIDINE WITH HEXAMETHYLENETETRAMINE AND WATER TO PROVIDE 4-(PYRIDIN-2-YL)BENZALDEHYDE SUMIKA FINE CHEMICALS CO., LTD. (JP) 2001-07-31 US disclosed
US-6242608-B1 REACTING 4-(PYRIDIN-2-YL)BENZALDEHYDE WITH HYDRAZINE TO FORM 4-(PYRIDIN-2-YL)BENZALDEHYDE HYDRAZONE; CHEMICAL INTERMEDIATE TO AN ANTI-HIV DRUG SUMIKA FINE CHEMICALS CO., LTD. (JP) 2001-06-05 US disclosed
US-6147218-A 2-phenylpyridine derivative and production method thereof SUMIKA FINE CHEMICALS CO., LTD. (JP) 2000-11-14 US disclosed
EP-0979820-A1 2-Phenylpyridine derivatives and production method thereof SUMIKA FINE CHEMICALS Co., Ltd. (JP) 2000-02-16 EP disclosed