SCHEMBL7057600

SCHEMBL7057600

O=C(O)Cc1ccc2c(c1)C(=O)c1ccccc1CC2

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 5/20 0.68
TDP1 Q9NUW8 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
CES1 P23141 1/20 0.50
HRH1 P35367 2/20 0.49
MAPK14 Q16539 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11088738 0.91 AKR1B1 (0.74) AKR1B1TDP1L3MBTL1CES1MAPK14
SCHEMBL16091063 0.91 AKR1B1 (0.63) AKR1B1HRH1
SCHEMBL16091078 0.85 AKR1B1 (0.67) AKR1B1
SCHEMBL14710258 0.83 AKR1B1 (0.61) AKR1B1TDP1MAPK14
SCHEMBL10922819 0.82 AKR1B1 (0.79) AKR1B1HRH1
SCHEMBL1347195 0.81 AKR1B1 (0.58) AKR1B1TDP1
SCHEMBL8600926 0.80 AKR1B1 (0.60) AKR1B1TDP1L3MBTL1
Isoxepac SCHEMBL24970 0.80 AKR1B1 (0.81) AKR1B1HRH1
SCHEMBL16091057 0.80 AKR1B1 (0.54) AKR1B1
Isoxepac SCHEMBL29588437 0.80 AKR1B1 (0.81) AKR1B1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042268-B1 1,7-DIBROMODIBENZOSUBERONE AND PROCEDURES FOR ITS PREPARATION BELUPO LIJEKOVI I KOZMETIKA D (HR) 2003-05-07 EP disclosed
EP-1042268-A1 DIBENZOSUBERONE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION Belupo - Lijekovi I Kozmetika D.O.O. (HR) 2000-10-11 EP disclosed
WO-1999028284-A1 DIBENZOSUBERONE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION BELUPO - LIJEKOVI I KOZMETIKA D.O.O. (HR) 1999-06-10 WO disclosed
US-4172949-A 2,4-Disubstituted-5-oxo-5H-dibenzo[a,d]cycloheptenes SYNTEX (U.S.A.) INC. (US) 1979-10-30 US disclosed
US-4020094-A ANTIINFLAMMATORY, ANALGESIC, ANTIPYRETIC SYNTEX (U.S.A.) INC. (US) 1977-04-26 US disclosed