SCHEMBL7068950

SCHEMBL7068950

CC(C)(C)OC(=O)NC(CC(=O)OCc1ccccc1)c1nc2ccccc2[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC10 Q969S8 1/20 0.54
HDAC11 Q96DB2 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HDAC9 Q9UKV0 1/20 0.54
HDAC5 Q9UQL6 1/20 0.54
AAK1 Q2M2I8 7/20 0.52
PTPN1 P18031 1/20 0.50
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
BCHE P06276 1/20 0.46
PPARA Q07869 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29095821 0.87 PPARA (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL24485487 0.87 PPARA (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL24143407 0.86 CYP1A2 (0.67) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL26304208 0.83 SCN10A (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8117254 0.83 HDAC3 (0.67) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL630992 0.82 PTPN1 (0.66) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2779366 0.81 AAK1 (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL15558774 0.81 MAPT (0.52) PPARAMAPTKLK7KLK5ALDH1A1
SCHEMBL9746641 0.80 AAK1 (0.68) AAK1PTPN1CYP3A4CYP2C9CYP2C19
SCHEMBL7299670 0.80 KLK5 (0.53) PPARAMAPTKLK7KLK5SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003062261-A2 DMT-TIC DI- AND TRI-PEPTIDIC DERIVATIVES AND RELATED COMPOSITIONS AND METHODS OF USE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2003-07-31 WO disclosed