SCHEMBL7077091

SCHEMBL7077091

C=CCc1cccc([N+](=O)[O-])c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.61
LMNA P02545 2/20 0.55
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
ALDH1A1 P00352 4/20 0.47
ACHE P22303 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ALOX15 P16050 1/20 0.47
MAPT P10636 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
POLB P06746 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PYCR1 P32322 1/20 0.47
PDE4A P27815 1/20 0.46
PDE4C Q08493 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formamide SCHEMBL28222941 0.94 TSHR (0.54) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL287236 0.85 TSHR (0.65) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL3718150 0.84 TSHR (0.62) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL9109568 0.83 TSHR (0.57) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL6158117 0.83 TSHR (0.57) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL16167547 0.83 TSHR (0.57) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL27554225 0.82 TSHR (0.61) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL28879992 0.82 TSHR (0.61) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL27456840 0.82 TSHR (0.61) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL28184209 0.82 TSHR (0.66) TSHRLMNACYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4587058-A Diisocyanates of the diphenyl methane series and processes for the production thereof BAYER AKTIENGESELLSCHAFT (DE) 1986-05-06 US claimed
EP-0046556-B1 DIISOCYANATES OR MIXTURES OF DIISOCYANATES OF THE DIPHENYLMETHANE CLASS, PROCESSES FOR THEIR PREPARATION, AS WELL AS THEIR USE AS SYNTHESIS COMPONENTS IN THE MANUFACTURE OF POLYURETHANES BY THE ISOCYANATE-POLYADDITION PROCESS BAYER AG (DE) 1983-03-09 EP claimed
EP-0046917-A1 Polyisocyanate mixtures of the diphenylmethane class, as well as their use as synthesis components in the manufacture of polyurethanes by the isocyanate-polyaddition process BAYER AG (DE) 1982-03-10 EP claimed
EP-0046556-A1 Diisocyanates or mixtures of diisocyanates of the diphenylmethane class, processes for their preparation, as well as their use as synthesis components in the manufacture of polyurethanes by the isocyanate-polyaddition process BAYER AG (DE) 1982-03-03 EP claimed
EP-1013636-B1 Preparation of allylic aromatic compounds AMERSHAM HEALTH AS (NO) 2003-07-09 EP disclosed
CN-1414951-A Drug discharge pump inhibitor FUNDAMENTAL THERAPEUTICAL INC (US) 2003-04-30 CN disclosed
US-6284894-B1 AROMATIC AMINE IS REACTED FIRST WITH A NITRITE AND THEN WITH AN ALLYLIC OLEFIN HAVING AN ELIMINATABLE TERMINAL SUBSTITUENT. NYCOMED IMAGING AS (NO) 2001-09-04 US disclosed
EP-1013636-A1 Preparation of allylic aromatic compounds NYCOMED IMAGING AS (NO) 2000-06-28 EP disclosed
CN-1087086-A Thiazolylvinylphenyl derivatives HOFFMANN LA ROCHE (CH) 1994-05-25 CN disclosed
US-5270309-A Kynurenic acid derivatives useful in the treatment of neurodegenerative disorders MERCK SHARP & DOHME LIMITED (GB) 1993-12-14 US disclosed
EP-0303387-B1 KYNURENIC ACID DERIVATIVES USEFUL IN THE TREATMENT OF NEURODEGENERATIVE DISORDERS MERCK SHARP & DOHME LTD. (GB) 1993-04-21 EP disclosed
EP-0303387-A1 Kynurenic acid derivatives useful in the treatment of neurodegenerative disorders MERCK SHARP & DOHME LTD. (GB) 1989-02-15 EP disclosed
US-4613687-A POLYURETHANES BAYER AKTIENGESELLSCHAFT (DE) 1986-09-23 US disclosed
US-4587058-A Diisocyanates of the diphenyl methane series and processes for the production thereof BAYER AKTIENGESELLSCHAFT (DE) 1986-05-06 US disclosed
EP-0046917-B1 POLYISOCYANATE MIXTURES OF THE DIPHENYLMETHANE CLASS, AS WELL AS THEIR USE AS SYNTHESIS COMPONENTS IN THE MANUFACTURE OF POLYURETHANES BY THE ISOCYANATE-POLYADDITION PROCESS BAYER AG (DE) 1983-12-07 EP disclosed
EP-0046556-B1 DIISOCYANATES OR MIXTURES OF DIISOCYANATES OF THE DIPHENYLMETHANE CLASS, PROCESSES FOR THEIR PREPARATION, AS WELL AS THEIR USE AS SYNTHESIS COMPONENTS IN THE MANUFACTURE OF POLYURETHANES BY THE ISOCYANATE-POLYADDITION PROCESS BAYER AG (DE) 1983-03-09 EP disclosed
EP-0046917-A1 Polyisocyanate mixtures of the diphenylmethane class, as well as their use as synthesis components in the manufacture of polyurethanes by the isocyanate-polyaddition process BAYER AG (DE) 1982-03-10 EP disclosed
EP-0046556-A1 Diisocyanates or mixtures of diisocyanates of the diphenylmethane class, processes for their preparation, as well as their use as synthesis components in the manufacture of polyurethanes by the isocyanate-polyaddition process BAYER AG (DE) 1982-03-03 EP disclosed