SCHEMBL7079031

SCHEMBL7079031

Nc1nc(NC2CCCCC2)nc(-c2ccc(O)cc2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.50
CSNK1D P48730 2/20 0.46
TPH1 P17752 1/20 0.44
BRAF P15056 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
ALOX5 P09917 2/20 0.41
HDAC1 Q13547 2/20 0.41
NUDT1 P36639 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
PDE5A O76074 1/20 0.40
ACP1 P24666 1/20 0.40
TYR P14679 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24342054 0.86 PDE5A (0.55) SMN1; SMN2HDAC1PDE5AACP1ADORA3
SCHEMBL19679830 0.86 PDE5A (0.55) SMN1; SMN2HDAC1PDE5AACP1ADORA3
SCHEMBL5336737 0.86 PDE5A (0.55) SMN1; SMN2HDAC1PDE5AACP1ADORA3
SCHEMBL22041442 0.86 PDE5A (0.55) SMN1; SMN2HDAC1PDE5AACP1ADORA3
SCHEMBL29117462 0.84 SMN1; SMN2 (0.48) SMN1; SMN2TPH1HDAC1PTGS1PTGS2
SCHEMBL29117417 0.84 NPSR1 (0.54) SMN1; SMN2HDAC1PDE5AACP1ADORA3
SCHEMBL29117406 0.81 NPC1 (0.59) SMN1; SMN2TPH1HDAC1NUDT1PTGS1
SCHEMBL29117468 0.81 SMN1; SMN2 (0.57) SMN1; SMN2CSNK1D
SCHEMBL29117469 0.78 NPC1 (0.59) SMN1; SMN2PDE4BPDE4D
SCHEMBL29117438 0.78 CHRNA7 (0.58) SMN1; SMN2PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030148269-A1 Centrifugally-enhanced method of determining ligand/target affinity HOLZMAN THOMAS F (US) 2003-08-07 US disclosed
EP-1161684-A1 CENTRIFUGALLY-ENHANCED METHOD OF DETERMINING LIGAND/TARGET AFFINITY ABBOTT LABORATORIES (US) 2001-12-12 EP disclosed
WO-2000055625-A1 CENTRIFUGALLY-ENHANCED METHOD OF DETERMINING LIGAND/TARGET AFFINITY ABBOTT LABORATORIES (US) 2000-09-21 WO disclosed