SCHEMBL7083274

SCHEMBL7083274

CC(=O)O[C@@H](CCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C1(c2ccccc2)CCC2(CC1)OCCO2

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 20/20 0.42
KCNH2 Q12809 1/20 0.42
SLC6A4 P31645 1/20 0.37
TACR3 P29371 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6492399 1.00 TACR1 (0.42) TACR1KCNH2SLC6A4TACR3
SCHEMBL6492394 1.00 TACR1 (0.42) TACR1KCNH2SLC6A4TACR3
SCHEMBL6484245 0.83 TACR1 (0.42) TACR1KCNH2SLC6A4
SCHEMBL6484240 0.83 TACR1 (0.42) TACR1KCNH2SLC6A4
SCHEMBL6492048 0.78 TACR1 (0.46) TACR1KCNH2SLC6A4TACR3
SCHEMBL6492051 0.78 TACR1 (0.46) TACR1KCNH2SLC6A4TACR3
SCHEMBL6485012 0.76 TACR1 (0.47) TACR1KCNH2SLC6A4
SCHEMBL6496791 0.72 TACR1 (0.43) TACR1KCNH2SLC6A4
SCHEMBL8923334 0.72 TACR1 (0.57) TACR1KCNH2SLC6A4
Hydrochloric Acid SCHEMBL8922068 0.71 TACR1 (0.56) TACR1KCNH2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286978-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2003-03-05 EP disclosed
WO-2001087866-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2001-11-22 WO disclosed