SCHEMBL7085228

SCHEMBL7085228

COC(=O)c1ccc(CCC2CC(OC)=CC(=O)O2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.70
ALDH1A1 P00352 3/20 0.61
TDP1 Q9NUW8 1/20 0.61
CYP4A11 Q02928 2/20 0.46
CYP4F2 P78329 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.42
IDH1 O75874 1/20 0.41
GRM2 Q14416 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2C19 P33261 2/20 0.40
HIF1A Q16665 2/20 0.40
TP53 P04637 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
ALOX12 P18054 1/20 0.40
CKS1B P61024 1/20 0.40
SKP2 Q13309 1/20 0.40
HSD17B10 Q99714 1/20 0.40
FAAH O00519 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18214442 0.86 CYP3A4 (0.76) CYP3A4ALDH1A1TDP1CYP1A2CYP2C19
SCHEMBL20148117 0.84 CYP3A4 (0.78) CYP3A4ALDH1A1TDP1CYP1A2CYP2C19
SCHEMBL18214373 0.83 CYP3A4 (0.76) CYP3A4ALDH1A1TDP1CYP1A2CYP2C19
SCHEMBL11308370 0.83 CYP3A4 (0.76) CYP3A4ALDH1A1TDP1GRM2CYP1A2
SCHEMBL5671273 0.83 CYP3A4 (0.76) CYP3A4ALDH1A1TDP1CYP1A2CYP2C19
SCHEMBL5671269 0.83 CYP3A4 (0.76) CYP3A4ALDH1A1TDP1CYP1A2CYP2C19
Dihydrokawain SCHEMBL2743647 0.83 CYP3A4 (1.00) CYP3A4ALDH1A1TDP1CYP1A2CYP2C19
SCHEMBL18214340 0.81 CYP3A4 (0.72) CYP3A4ALDH1A1TDP1CYP1A2CYP2C19
SCHEMBL12371088 0.81 CYP4A11 (0.49) CYP3A4ALDH1A1CYP4A11CYP4F2LOXL2
SCHEMBL18214367 0.80 CYP3A4 (0.70) CYP3A4ALDH1A1TDP1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030236302-A1 Synthetic derivatives SYNTA PHARMACEUTICALS CORP. 2003-12-25 US disclosed
WO-2003072103-A1 SYNTHETIC DERIVATIVES KAVA PHARMACEUTICALS, INC. (US) 2003-09-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030236302-A1 Synthetic derivatives CBR1, CBR3, REL CYP3A4 169/4885ALDH1A1 1421/4885TDP1 3358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.