SCHEMBL7085656

SCHEMBL7085656

CCCCCCCN1CC[C@@H](COc2ccnc3ccc(OC)cc23)[C@@H](CC)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 2/20 0.53
CYP2D6 P10635 4/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
HSD17B10 Q99714 3/20 0.43
KCNH2 Q12809 3/20 0.43
TSHR P16473 1/20 0.43
MEN1 O00255 1/20 0.43
CYP3A4 P08684 1/20 0.43
KMT2A Q03164 1/20 0.43
CHRM2 P08172 1/20 0.43
ADRA2A P08913 1/20 0.43
SLC6A4 P31645 1/20 0.43
OPRM1 P35372 1/20 0.43
SLC6A3 Q01959 1/20 0.43
SLC2A1 P11166 1/20 0.40
HTR1A P08908 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974309 0.86 CCR8 (0.57) CCR8KCNH2SLC2A1HTR1AADRA1D
SCHEMBL6965276 0.85 CCR8 (0.53) CCR8CYP2D6KDM4EALDH1A1HPGD
SCHEMBL6971729 0.84 CCR8 (0.52) CCR8CYP2D6KDM4EALDH1A1HPGD
SCHEMBL6968481 0.83 CCR8 (0.49) CCR8CYP2D6KDM4EALDH1A1HPGD
SCHEMBL6977734 0.82 CCR8 (0.51) CCR8CYP2D6KDM4EALDH1A1HPGD
SCHEMBL6969955 0.82 CCR8 (0.51) CCR8CYP2D6KDM4EALDH1A1HPGD
SCHEMBL6968986 0.82 CCR8 (0.51) CCR8CYP2D6KDM4EALDH1A1HPGD
SCHEMBL6968990 0.82 CCR8 (0.51) CCR8CYP2D6KDM4EALDH1A1HPGD
SCHEMBL8127825 0.82 CCR8 (0.53) CCR8KCNH2SLC6A4SLC2A1ADRA1B
SCHEMBL6975290 0.82 KCNH2 (0.56) CYP2D6KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051413-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-06-04 EP claimed