SCHEMBL7085946

SCHEMBL7085946

CC#CC[C@@H](CCC)C(=O)NCCC(C)CC(N)=O

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC7 Q8WUI4 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC9 Q9UKV0 2/20 0.36
HDAC5 Q9UQL6 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
ECE1 P42892 1/20 0.34
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
TSHR P16473 2/20 0.33
USP2 O75604 2/20 0.33
GRIK1 P39086 1/20 0.33
GRIK2 Q13002 1/20 0.33
DPP7 Q9UHL4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085943 0.88 GRIK1 (0.34) HDAC7HDAC8HDAC6HDAC9HDAC5
SCHEMBL7082813 0.80 GRIK1 (0.38) HDAC7HDAC8HDAC6HDAC9HDAC5
SCHEMBL7081675 0.73 GRIK1 (0.37) HDAC7HDAC8HDAC6HDAC9HDAC5
SCHEMBL7134376 0.73 GRIK1 (0.37) HDAC7HDAC8HDAC6HDAC9HDAC5
SCHEMBL7085892 0.71 GRIK1 (0.46) HDAC7HDAC8HDAC6HDAC9HDAC5
SCHEMBL7082795 0.71 GRIK1 (0.46) HDAC7HDAC8HDAC6HDAC9HDAC5
SCHEMBL7085940 0.71 GRIK1 (0.36) HDAC7HDAC8HDAC6HDAC9HDAC5
SCHEMBL7085945 0.70 ERAP2 (0.40) HDAC8HDAC3HDAC4HDAC1HDAC2
SCHEMBL25078569 0.69
SCHEMBL276380 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1330429-A2 ALKYNYL AMIDES AND THEIR THERAPEUTIC APPLICATIONS Abbott Laboratories (US) 2003-07-30 EP claimed
WO-2002036546-A2 ALKYNYL AMIDES AND THEIR THERAPEUTIC APPLICATIONS ABBOTT LABORATORIES (US) 2002-05-10 WO claimed
EP-1330429-A2 ALKYNYL AMIDES AND THEIR THERAPEUTIC APPLICATIONS Abbott Laboratories (US) 2003-07-30 EP disclosed
WO-2002036546-A2 ALKYNYL AMIDES AND THEIR THERAPEUTIC APPLICATIONS ABBOTT LABORATORIES (US) 2002-05-10 WO disclosed