SCHEMBL7086777

SCHEMBL7086777

COC(=O)c1ccc(C=O)cc1.COC(=O)c1ccc(CNc2cc(-c3cc4cc(F)c(F)cc4[nH]3)ccc2OC)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.39
ALDH1A1 P00352 3/20 0.39
HPSE Q9Y251 2/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALOX15 P16050 1/20 0.36
ERN1 O75460 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6494687 0.94 HDAC8 (0.44) HDAC8ALDH1A1HPSEHDAC1HDAC6
SCHEMBL6493899 0.82 MAPT (0.47) ALDH1A1SMN1; SMN2KDM4ELMNAMAPT
SCHEMBL6492806 0.80 KMT2A (0.40) SMN1; SMN2KDM4ELMNAMAPTHPGD
Hydrochloric Acid SCHEMBL6493224 0.79 KMT2A (0.39) SMN1; SMN2KDM4EMAPTHPGDKMT2A
SCHEMBL6493106 0.79 MAPT (0.54) ALDH1A1SMN1; SMN2KDM4ELMNAMAPT
SCHEMBL6496748 0.78 PI4KB (0.42) ALDH1A1SMN1; SMN2KDM4ELMNAMAPT
SCHEMBL7073827 0.78 MAPT (0.41) ALDH1A1HPSESMN1; SMN2KDM4ELMNA
Hydrochloric Acid SCHEMBL7073825 0.77 MAPT (0.41) ALDH1A1HPSESMN1; SMN2KDM4ELMNA
SCHEMBL6496194 0.77 MAPT (0.43) HDAC8ALDH1A1HDAC1HDAC6SMN1; SMN2
SCHEMBL6503258 0.75 ABCB1 (0.46) ALDH1A1SMN1; SMN2KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294686-A2 INDOLE DERIVATIVES AND THEIR USE AS 15-LIPOXYGENASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2003-03-26 EP disclosed
WO-2001096299-A2 INDOLE DERIVATIVES AND THEIR USE AS 15-LIPOXYGENASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-12-20 WO disclosed