SCHEMBL7090134

SCHEMBL7090134

COc1cc(OC)c(OC)cc1CCCO

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TNKS2 Q9H2K2 1/20 0.50
CYP3A4 P08684 1/20 0.50
HTR2A P28223 5/20 0.49
CYP19A1 P11511 1/20 0.49
TAAR1 Q96RJ0 4/20 0.46
HMGCR P04035 1/20 0.46
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
HTR2C P28335 1/20 0.43
GLA P06280 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581243 0.92 HTR2A (0.49) TNKS2CYP3A4HTR2ACYP19A1TAAR1
SCHEMBL580783 0.92 HTR2A (0.49) TNKS2CYP3A4HTR2ACYP19A1TAAR1
SCHEMBL580350 0.92 HTR2A (0.49) TNKS2CYP3A4HTR2ACYP19A1TAAR1
SCHEMBL580254 0.92 HTR2A (0.49) TNKS2CYP3A4HTR2ACYP19A1TAAR1
SCHEMBL580817 0.92 HTR2A (0.49) TNKS2CYP3A4HTR2ACYP19A1TAAR1
SCHEMBL31265265 0.82 SMN1; SMN2 (0.50) TNKS2HTR2ATAAR1HMGCRPDE4A
SCHEMBL31295158 0.82 TNKS2 (0.46) TNKS2HTR2ATAAR1HMGCRHTR2C
SCHEMBL21798808 0.82 TAAR1 (0.52) TNKS2CYP3A4HTR2ACYP19A1TAAR1
SCHEMBL5304175 0.81 HTR2A (0.70) HTR2ATAAR1HTR2C
SCHEMBL5304173 0.81 HTR2A (0.70) HTR2ATAAR1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102199077-B Method for producing (E)-2,4,5-trimethoxy-1-propenylbenzene LU CHAO 2013-01-23 CN claimed
CN-102199077-A Method for producing (E)-2,4,5-trimethoxy-1-propenylbenzene CHAO LU 2011-09-28 CN claimed
CN-101195562-A Novel method for synthesizing alpha-asarone GUANGXI TRADITIONAL CHINESE ME (CN) 2008-06-11 CN claimed
WO-2003082786-A1 A PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE ALPHA-ASARONE FROM TOXIC BETA-ASARONE RICH ACORUS CALAMUS OIL COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2003-10-09 WO claimed
CN-102199077-B Method for producing (E)-2,4,5-trimethoxy-1-propenylbenzene LU CHAO 2013-01-23 CN disclosed
CN-102199077-A Method for producing (E)-2,4,5-trimethoxy-1-propenylbenzene CHAO LU 2011-09-28 CN disclosed
CN-101492351-A Process for producing asarin YABANG CHEMICAL INDUSTRY GROUP (CN) 2009-07-29 CN disclosed
CN-101195562-A Novel method for synthesizing alpha-asarone GUANGXI TRADITIONAL CHINESE ME (CN) 2008-06-11 CN disclosed
WO-2003082786-A1 A PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE ALPHA-ASARONE FROM TOXIC BETA-ASARONE RICH ACORUS CALAMUS OIL COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2003-10-09 WO disclosed
WO-2003082786-A1 A PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE ALPHA-ASARONE FROM TOXIC BETA-ASARONE RICH ACORUS CALAMUS OIL COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2003-10-09 WO disclosed
US-6590127-B1 Formation of alpha-asarone, isoacoramone and 2,4,5-trimethoxycinnamaldehyde in one step process via 2,3-dichloro-5,6-dicyano-1,4-benzoquinone assisted dehydrogenation/oxidation of 2,4,5-trimethoxyphenylpropane COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2003-07-08 US disclosed
US-6590127-B1 Formation of alpha-asarone, isoacoramone and 2,4,5-trimethoxycinnamaldehyde in one step process via 2,3-dichloro-5,6-dicyano-1,4-benzoquinone assisted dehydrogenation/oxidation of 2,4,5-trimethoxyphenylpropane COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2003-07-08 US disclosed