SCHEMBL7090213

SCHEMBL7090213

O=C(O)C1CCN(c2cc(N3CCN(C(=O)N(c4ccccc4)C(F)(F)F)CC3)c([N+](=O)[O-])cc2C(F)(F)F)CC1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 11/20 0.65
TDP1 Q9NUW8 1/20 0.47
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
POLB P06746 1/20 0.46
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
FFAR2 O15552 1/20 0.43
GPR174 Q9BXC1 3/20 0.42
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089371 0.84 SERPINE1 (0.72) SERPINE1TDP1CYP2C9CYP2C19POLB
SCHEMBL7087924 0.81 SERPINE1 (0.75) SERPINE1TDP1CYP2C9CYP2C19POLB
SCHEMBL7084123 0.79 SERPINE1 (0.82) SERPINE1TDP1CYP2C9CYP2C19POLB
SCHEMBL7088169 0.79 SERPINE1 (1.00) SERPINE1TDP1CYP2C9CYP2C19POLB
SCHEMBL7091396 0.78 SERPINE1 (1.00) SERPINE1MAPT
SCHEMBL7087964 0.77 SERPINE1 (1.00) SERPINE1CYP2C9CYP2C19POLBMAPT
SCHEMBL7085406 0.75 SERPINE1 (0.77) SERPINE1MAPT
SCHEMBL7084622 0.75 SERPINE1 (1.00) SERPINE1TDP1CYP2C9CYP2C19POLB
SCHEMBL7084109 0.75 SERPINE1 (0.82) SERPINE1TDP1CYP2C9CYP2C19POLB
SCHEMBL7165057 0.75 SERPINE1 (1.00) SERPINE1TDP1CYP2C9CYP2C19POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003080060-A1 SUBSTITUTED PIPERAZINE ANTITHROMBOTIC PAI-1 INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2003-10-02 WO disclosed